![Discovery of Small Molecule Kappa Opioid Receptor Agonist and Antagonist Chemotypes through a HTS and Hit Refinement Strategy]()
Discovery of Small Molecule Kappa Opioid Receptor Agonist and Antagonist Chemotypes through a HTS and Hit Refinement StrategyFrankowski, Kevin J.; Hedrick, Michael P.; Gosalia, Palak; Li, Kelin; Shi, Shenghua; Whipple, David; Ghosh, Partha; Prisinzano, Thomas E.; Schoenen, Frank J.; Su, Ying; Vasile, S.; Sergienko, Eduard; Gray, Wilson; Hariharan, Santosh; Milan, Loribelle; Heynen-Genel, Susanne; Mangravita-Novo, Arianna; Vicchiarelli, Michael; Smith, Layton H.; Streicher, John M.; Caron, Marc G.; Barak, Lawrence S.; Bohn, Laura M.; Chung, Thomas D. Y.; Aubé, Jeffrey · ACS Chemical Neuroscience · 2012