Design and synthesis of conformationally-constrained MMP inhibitors
- 作者Michael G. Natchus; Menyan Cheng; Christopher T. Wahl; Stanislaw Pikul; Neil G. Almstead; Rimma S. Bradley; Yetunde O. Taiwo; Glen E. Mieling; C.Michelle Dunaway; Catherine E. Snider; John M. McIver; Bobby L. Barnett; Sara J. McPhail; Melanie B. Anastasio; Biswanath De
- 卷第8卷
- 期第16期
- 印刷ISSN0960-894X
- 文件大小271.77KB
- 发表时间1998
- DOI10.1016/s0960-894x(98)00370-9
- 页码2077-2080
Peptidyl human heart chymase inhibitors. 1. Synthesis and inhibitory activity of difluoromethylene ketone derivatives bearing P′ binding subsitesMasahiro Eda; Atsuyuki Ashimori; Fumihiko Akahoshi; Takuya Yoshimura; Yoshihisa Inoue; Chikara Fukaya; Masahide Nakajima; Hajime Fukuyama; Teruaki Imada; Norifumi Nakamura · 1998
Peptidyl human heart chymase inhibitors. 2. Discovery of highly selective difluoromethylene ketone derivatives with Glu AT P3 siteMasahiro Eda; Atsuyuki Ashimori; Fumihiko Akahoshi; Takuya Yoshimura; Yoshihisa Inoue; Chikara Fukaya; Masahide Nakajima; Hajime Fukuyama; Teruaki Imada; Norifumi Nakamura · 1998
Corrigendum to “Peptidyl human heart chymase inhibitors. Part 1: Synthesis and inhibitory activity of difluoromethylene ketone derivatives bearing P′ binding subsites” [Bioorg. Med. Chem. Lett. 8 (1998) 913]Masahiro Eda; Atsuyuki Ashimori; Fumihiko Akahoshi; Takuya Yoshimura; Yoshihisa Inoue; Chikara Fukaya; Masahide Nakajima; Hajime Fukuyama; Teruaki Imada; Norifumi Nakamura · 1998