Discovery of 4-heteroarylbicyclo[2.2.2]octyltriazoles as potent and selective inhibitors of 11β-HSD1: Novel therapeutic agents for the treatment of metabolic syndrome
Xin Gu; Jasminka Dragovic; Gloria C. Koo; Sam L. Koprak; Cheryl LeGrand; Steven S. Mundt; Kashmira Shah; Marty S. Springer; Eugene Y. Tan; Rolf Thieringer; Anne Hermanowski-Vosatka; Hratch J. Zokian; James M. Balkovec; Sherman T. Waddell
- 作者Xin Gu; Jasminka Dragovic; Gloria C. Koo; Sam L. Koprak; Cheryl LeGrand; Steven S. Mundt; Kashmira Shah; Marty S. Springer; Eugene Y. Tan; Rolf Thieringer; Anne Hermanowski-Vosatka; Hratch J. Zokian; James M. Balkovec; Sherman T. Waddell
- 卷第15卷
- 期第23期
- 印刷ISSN0960-894X
- 文件大小126.88KB
- 发表时间2005
- DOI10.1016/j.bmcl.2005.08.052
- 页码5266-5269