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Optimization of a pyrazoloquinolinone class of Chk1 kinase inhibitors

Optimization of a pyrazoloquinolinone class of Chk1 kinase inhibitors

Edward J. Brnardic; Robert M. Garbaccio; Mark E. Fraley; Edward S. Tasber; Justin T. Steen; Kenneth L. Arrington; Vadim Y. Dudkin; George D. Hartman; Steven M. Stirdivant; Bob A. Drakas; Keith Rickert; Eileen S. Walsh; Kelly Hamilton; Carolyn A. Buser; James Hardwick; Weikang Tao; Stephen C. Beck; Xianzhi Mao; Robert B. Lobell; Laura Sepp-Lorenzino; Youwei Yan; Mari Ikuta; Sanjeev K. Munshi; Lawrence C. Kuo; Constantine Kreatsoulas
  • 作者Edward J. Brnardic; Robert M. Garbaccio; Mark E. Fraley; Edward S. Tasber; Justin T. Steen; Kenneth L. Arrington; Vadim Y. Dudkin; George D. Hartman; Steven M. Stirdivant; Bob A. Drakas; Keith Rickert; Eileen S. Walsh; Kelly Hamilton; Carolyn A. Buser; James Hardwick; Weikang Tao; Stephen C. Beck; Xianzhi Mao; Robert B. Lobell; Laura Sepp-Lorenzino; Youwei Yan; Mari Ikuta; Sanjeev K. Munshi; Lawrence C. Kuo; Constantine Kreatsoulas
  • 卷第17卷
  • 期第21期
  • 印刷ISSN0960-894X
  • 文件大小465.86KB
  • 发表时间2007
  • DOI10.1016/j.bmcl.2007.07.051
  • 页码5989-5994
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