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CCR5 inhibitors: emergence, success, and challengesMaeda, Kenji; Das, Debananda; Nakata, Hirotomo; Mitsuya, Hiroaki · Expert Opinion on Emerging Drugs · 2012
Discovery of orally available spirodiketopiperazine-based CCR5 antagonistsRena Nishizawa; Toshihiko Nishiyama; Katsuya Hisaichi; Keisuke Hirai; Hiromu Habashita; Yoshikazu Takaoka; Hideaki Tada; Kenji Sagawa; Shiro Shibayama; Kenji Maeda; Hiroaki Mitsuya; Hisao Nakai; Daikichi Fukushima; Masaaki Toda · 2010
Spirodiketopiperazine-based CCR5 antagonists: Improvement of their pharmacokinetic profilesRena Nishizawa; Toshihiko Nishiyama; Katsuya Hisaichi; Keisuke Hirai; Hiromu Habashita; Yoshikazu Takaoka; Hideaki Tada; Kenji Sagawa; Shiro Shibayama; Kenji Maeda; Hiroaki Mitsuya; Hisao Nakai; Daikichi Fukushima; Masaaki Toda · 2010
Spirodiketopiperazine-based CCR5 antagonists: Lead optimization from biologically active metaboliteRena Nishizawa; Toshihiko Nishiyama; Katsuya Hisaichi; Naoki Matsunaga; Chiaki Minamoto; Hiromu Habashita; Yoshikazu Takaoka; Masaaki Toda; Shiro Shibayama; Hideaki Tada; Kenji Sagawa; Daikichi Fukushima; Kenji Maeda; Hiroaki Mitsuya · 2007
Spirodiketopiperazine-based CCR5 antagonist: Discovery of an antiretroviral drug candidateRena Nishizawa; Toshihiko Nishiyama; Katsuya Hisaichi; Chiaki Minamoto; Naoki Matsunaga; Yoshikazu Takaoka; Hisao Nakai; Stephen Jenkinson; Wieslaw M. Kazmierski; Hideaki Tada; Kenji Sagawa; Shiro Shibayama; Daikichi Fukushima; Kenji Maeda; Hiroaki Mitsuya · 2011
Design and synthesis of novel HIV-1 protease inhibitors incorporating oxyindoles as the -ligandsArun K. Ghosh; Gary Schiltz; Ramu Sridhar Perali; Sofiya Leshchenko; Stephanie Kay; D. Eric Walters; Yasuhiro Koh; Kenji Maeda; Hiroaki Mitsuya · 2006
Design and Synthesis of Novel HIV-1 Protease Inhibitors Incorporating Oxyindoles as the P2′-Ligands.Arun K. Ghosh; Gary Schiltz; Ramu Sridhar Perali; Sofiya Leshchenko; Stephanie Kay; D. Eric Walters; Yasuhiro Koh; Kenji Maeda; Hiroaki Mitsuya · 2006