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Exploration and optimization of substituted triazolothiadiazines and triazolopyridazines as PDE4 inhibitors

Exploration and optimization of substituted triazolothiadiazines and triazolopyridazines as PDE4 inhibitors

Amanda P. Skoumbourdis; Christopher A. LeClair; Eduard Stefan; Adrian G. Turjanski; William Maguire; Steven A. Titus; Ruili Huang; Douglas S. Auld; James Inglese; Christopher P. Austin; Stephen W. Michnick; Menghang Xia; Craig J. Thomas
  • 作者Amanda P. Skoumbourdis; Christopher A. LeClair; Eduard Stefan; Adrian G. Turjanski; William Maguire; Steven A. Titus; Ruili Huang; Douglas S. Auld; James Inglese; Christopher P. Austin; Stephen W. Michnick; Menghang Xia; Craig J. Thomas
  • 卷第19卷
  • 期第13期
  • 印刷ISSN0960-894X
  • 文件大小577.74KB
  • 发表时间2009
  • DOI10.1016/j.bmcl.2009.01.057
  • 页码3686-3692
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