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Discovery and structure–activity relationships of a series of pyroglutamic acid amide antagonists of the P2X7 receptor

Discovery and structure–activity relationships of a series of pyroglutamic acid amide antagonists of the P2X7 receptor

Muna H. Abdi; Paul J. Beswick; Andy Billinton; Laura J. Chambers; Andrew Charlton; Sue D. Collins; Katharine L. Collis; David K. Dean; Elena Fonfria; Robert J. Gleave; Clarisse L. Lejeune; David G. Livermore; Stephen J. Medhurst; Anton D. Michel; Andrew P. Moses; Lee Page; Sadhana Patel; Shilina A. Roman; Stefan Senger; Brian Slingsby; Jon G.A. Steadman; Alexander J. Stevens; Daryl S. Walter
  • 作者Muna H. Abdi; Paul J. Beswick; Andy Billinton; Laura J. Chambers; Andrew Charlton; Sue D. Collins; Katharine L. Collis; David K. Dean; Elena Fonfria; Robert J. Gleave; Clarisse L. Lejeune; David G. Livermore; Stephen J. Medhurst; Anton D. Michel; Andrew P. Moses; Lee Page; Sadhana Patel; Shilina A. Roman; Stefan Senger; Brian Slingsby; Jon G.A. Steadman; Alexander J. Stevens; Daryl S. Walter
  • 卷第20卷
  • 期第17期
  • 印刷ISSN0960-894X
  • 文件大小720.30KB
  • 发表时间2010
  • DOI10.1016/j.bmcl.2010.07.033
  • 页码5080-5084
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