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Discovery of a potent and selective Bcl-2 inhibitor using SAR by NMR

Discovery of a potent and selective Bcl-2 inhibitor using SAR by NMR

Andrew M. Petros; Jeffrey R. Huth; Thorsten Oost; Cheol-Min Park; Hong Ding; Xilu Wang; Haichao Zhang; Paul Nimmer; Renaldo Mendoza; Chaohong Sun; Jamey Mack; Karl Walter; Sarah Dorwin; Emily Gramling; Uri Ladror; Saul H. Rosenberg; Steven W. Elmore; Stephen W. Fesik; Philip J. Hajduk
  • 作者Andrew M. Petros; Jeffrey R. Huth; Thorsten Oost; Cheol-Min Park; Hong Ding; Xilu Wang; Haichao Zhang; Paul Nimmer; Renaldo Mendoza; Chaohong Sun; Jamey Mack; Karl Walter; Sarah Dorwin; Emily Gramling; Uri Ladror; Saul H. Rosenberg; Steven W. Elmore; Stephen W. Fesik; Philip J. Hajduk
  • 卷第20卷
  • 期第22期
  • 印刷ISSN0960-894X
  • 文件大小1880.29KB
  • 发表时间2010
  • DOI10.1016/j.bmcl.2010.09.033
  • 页码6587-6591
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