Pyrrolo[1,2-f]triazines as JAK2 inhibitors: Achieving potency and selectivity for JAK2 over JAK3
Lalgudi S. Harikrishnan; Muthoni G. Kamau; Honghe Wan; Jennifer A. Inghrim; Kurt Zimmermann; Xiaopeng Sang; Harold A. Mastalerz; Walter L. Johnson; Guifen Zhang; Louis J. Lombardo; Michael A. Poss; George L. Trainor; John S. Tokarski; Matthew V. Lorenzi; Dan You; Marco M. Gottardis; Kathy F. Baldwin; Jonathan Lippy; David S. Nirschl; Ruhui Qiu; Arthur V. Miller; Javed Khan; John S. Sack; Ashok V. Purandare
- 作者Lalgudi S. Harikrishnan; Muthoni G. Kamau; Honghe Wan; Jennifer A. Inghrim; Kurt Zimmermann; Xiaopeng Sang; Harold A. Mastalerz; Walter L. Johnson; Guifen Zhang; Louis J. Lombardo; Michael A. Poss; George L. Trainor; John S. Tokarski; Matthew V. Lorenzi; Dan You; Marco M. Gottardis; Kathy F. Baldwin; Jonathan Lippy; David S. Nirschl; Ruhui Qiu; Arthur V. Miller; Javed Khan; John S. Sack; Ashok V. Purandare
- 卷第21卷
- 期第5期
- 印刷ISSN0960-894X
- 文件大小902.70KB
- 发表时间2011
- DOI10.1016/j.bmcl.2011.01.022
- 页码1425-1428