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Identification of a Conformational Equilibrium That Determines the Efficacy and Functional Selectivity of the μ-Opioid Receptor

Identification of a Conformational Equilibrium That Determines the Efficacy and Functional Selectivity of the μ-Opioid Receptor

Okude, Junya; Ueda, Takumi; Kofuku, Yutaka; Sato, Motohiko; Nobuyama, Naoyuki; Kondo, Keita; Shiraishi, Yutaro; Mizumura, Takuya; Onishi, Kento; Natsume, Mei; Maeda, Masahiro; Tsujishita, Hideki; Kuranaga, Takefumi; Inoue, Masayuki; Shimada, Ichio
  • 期刊名称Angewandte Chemie International Edition
  • 作者Okude, Junya; Ueda, Takumi; Kofuku, Yutaka; Sato, Motohiko; Nobuyama, Naoyuki; Kondo, Keita; Shiraishi, Yutaro; Mizumura, Takuya; Onishi, Kento; Natsume, Mei; Maeda, Masahiro; Tsujishita, Hideki; Kuranaga, Takefumi; Inoue, Masayuki; Shimada, Ichio
  • 卷第54卷
  • 期第52期
  • 印刷ISSN1433-7851
  • 文件大小2932.58KB
  • 发表时间2015-12-21
  • DOI10.1002/anie.201508794
  • 页码15771-15776
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