TAS4464, a highly potent and selective inhibitor of NEDD8 activating enzyme, suppresses neddylation and shows antitumor activity in diverse cancer models
Yoshimura, Chihoko; Muraoka, Hiromi; Ochiiwa, Hiroaki; Tsuji, Shingo; Hashimoto, Akihiro; Kazuno, Hiromi; Nakagawa, Fumio; Komiya, Yu; Suzuki, Satoshi; Takenaka, Toru; Kumazaki, Masafumi; Fujita, Naoya; Mizutani, Takashi; Ohkubo, Shuichi
- 期刊名称Molecular Cancer Therapeutics
- 作者Yoshimura, Chihoko; Muraoka, Hiromi; Ochiiwa, Hiroaki; Tsuji, Shingo; Hashimoto, Akihiro; Kazuno, Hiromi; Nakagawa, Fumio; Komiya, Yu; Suzuki, Satoshi; Takenaka, Toru; Kumazaki, Masafumi; Fujita, Naoya; Mizutani, Takashi; Ohkubo, Shuichi
- 印刷ISSN1535-7163
- 电子ISSN1538-8514
- 文件大小1493.34KB
- 发表时间2019-05-15
- DOI10.1158/1535-7163.MCT-18-0644