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Discovery of (2
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-indol-7-yl]-2-(4-methylpiperazin-1-yl)propenamide (AZD4205) as a Potent and Selective Janus Kinase 1 InhibitorSu, Qibin; Banks, Erica; Bebernitz, Geraldine; Bell, Kirsten; Borenstein, Cassandra F.; Chen, Huawei; Chuaqui, Claudio E.; Deng, Nanhua; Ferguson, Andrew D.; Kawatkar, Sameer; Grimster, Neil P.; Ruston, Linette; Lyne, Paul D.; Read, Jon A.; Peng, Xianyou; Pei, Xiaohui; Fawell, Stephen; Tang, Zhanlei; Throner, Scott; Vasbinder, Melissa M.; Wang, Haoyu; Winter-Holt, Jon; Woessner, Richard; Wu, Allan; Yang, Wenzhan; Zinda, Michael; Kettle, Jason G. · Journal of Medicinal Chemistry · 2020