Lewis acid control of asymmetric synthesis
- 作者Keiji Maruoka
- 卷第57卷
- 期第5期
- 印刷ISSN0040-4020
- 文件大小35.75KB
- 发表时间2001
- DOI10.1016/s0040-4020(00)01037-1
ChemInform Abstract: Diastereoselective Synthesis of the Acid Part of a New Muscarinic M3 Receptor Antagonist.Morihiro Mitsuya; Yoshio Ogino; Norikazu Ohtake; Toshiaki Mase · 2001
J-104129, a novel muscarinic M3 receptor antagonist with high selectivity for M3 over M2 receptorsMorihiro Mitsuya; Toshiaki Mase; Yoshimi Tsuchiya; Kumiko Kawakami; Hiromi Hattori; Kensuke Kobayashi; Yoshio Ogino; Toru Fujikawa; Akio Satoh; Toshifumi Kimura; Kazuhito Noguchi; Norikazu Ohtake; Koji Tomimoto · 1999
Discovery of 2-Aminothiazole-4-carboxamides, a Novel Class of Muscarinic M3 Selective Antagonists, Through Solution-Phase Parallel Synthesis.Yufu Sagara; Morihiro Mitsuya; Minaho Uchiyama; Yoshio Ogino; Toshifumi Kimura; Norikazu Ohtake; Toshiaki Mase · 2005
Discovery of 2-Aminothiazole-4-carboxamides, a Novel Class of Muscarinic M3 Selective Antagonists, through Solution-Phase Parallel SynthesisSagara, Yufu; Mitsuya, Morihiro; Uchiyama, Minaho; Ogino, Yoshio; Kimura, Toshifumi; Ohtake, Norikazu; Mase, Toshiaki · CHEMICAL & PHARMACEUTICAL BULLETIN · 2005
Discovery of a muscarinic M3 receptor antagonist with high selectivity for M3 over M2 receptors among 2-[(1S,3S)-3-sulfonylaminocyclopentyl]phenylacetamide derivativesMorihiro Mitsuya; Yoshio Ogino; Kumiko Kawakami; Minaho Uchiyama; Toshifumi Kimura; Tomoshige Numazawa; Takuro Hasegawa; Norikazu Ohtake; Kazuhito Noguchi; Toshiaki Mase · 2000
A Potent, Long-Acting, Orally Active (2 <i>R</i> )-2-[(1 <i>R</i> )-3,3-Difluorocyclopentyl]-2-hydroxy-2-phenylacetamide: A Novel Muscarinic M <sub/>3</sub> Receptor Antagonist with High Selectivity for M <sub/>3</sub> over M <sub/>2</sub> ReceptorsMitsuya, Morihiro; Kobayashi, Kensuke; Kawakami, Kumiko; Satoh, Atsushi; Ogino, Yoshio; Kakikawa, Taro; Ohtake, Norikazu; Kimura, Toshifumi; Hirose, Hiroyasu; Sato, Akio; Numazawa, Tomosige; Hasegawa, Takuro; Noguchi, Kazuhito; Mase, Toshiaki · Journal of Medicinal Chemistry · 2000