![Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit]()
Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment HitGerstenberger, Brian S.; Trzupek, John D.; Tallant, Cynthia; Fedorov, Oleg; Filippakopoulos, Panagis; Brennan, Paul E.; Fedele, Vita; Martin, Sarah; Picaud, Sarah; Rogers, Catherine; Parikh, Mihir; Taylor, Alexandria; Samas, Brian; O’Mahony, Alison; Berg, Ellen; Pallares, Gabriel; Torrey, Adam D.; Treiber, Daniel K.; Samardjiev, Ivan J.; Nasipak, Brian T.; Padilla-Benavides, Teresita; Wu, Qiong; Imbalzano, Anthony N.; Nickerson, Jeffrey A.; Bunnage, Mark E.; Müller, Susanne; Knapp, Stefan; Owen, Dafydd R. · Journal of Medicinal Chemistry · 2016